GIP (native; Selective Acyl-GIP / CNS-Gipr-KO)
MARKETED
CNS-GIPR signalling regulates body weight and food intake: HFD-fed CNS-Gipr-KO and humanised-GIPR mice with CNS-hGIPR deletion show decreased body weight, and acute...
Zhang Q et al., Cell Metab 2021;33(4):833-844.e5
Source
Full findingCNS-GIPR signalling regulates body weight and food intake: HFD-fed CNS-Gipr-KO and humanised-GIPR mice with CNS-hGIPR deletion show decreased body weight, and acute central/peripheral acyl-GIP raises cFos in hypothalamic feeding centres coinciding with decreased food intake; the GLP-1/GIP co-agonist intake advantage is extinguished in CNS-Gipr-KO. This is the CNS-GIP appetite-suppression pole.
PopulationMice (genetic + acyl-GIP)
Fundingacademic/independent analysis (manufacturer not study sponsor; per-study COI not individually audited)
Scope limitsReused from corpus T9-GIPR-01. AGONISM pole of the GIP agonism-vs-antagonism appetite paradox. Mouse — does not license a human CNS-GIP-appetite attribution.
Comparatorsvehicle; GLP-1/GIP co-agonist